Product Overview
(-)-Indolactam V | T17299 | TargetMol Chemicals
CAS: 90365-57-4
Smiles: CC(C)[C@@H]1N(C)c2cccc3[nH]cc(C[C@@H](CO)NC1=O)c23
Formula: C17H23N3O2
Pathway: Chromatin/Epigenetic|||Cytoskeletal Signaling
Target: PKC
Receptor: N/A
Bioactivity: (-)-Indolactam V is a PKC activator (Kis: 3.36 nM, 1.03 μM for η-CRD2, γ-CRD2). (-)-Indolactam V also has the Kds are 5.5 nM (η-C1B), 7.7 nM (ε-C1B), 8.3 nM (δ-C1B), 18.9 nM (β-C1A-long), 20.8 nM (α-C1A-long), 137 nM (β-C1B), 138 nM (γ-C1A), 213 nM (γ-C1B). It has antitumor activity.
Molecular Weight: 301, 39
