Product Overview
Islatravir | T16098 | TargetMol Chemicals
CAS: 865363-93-5
Smiles: Nc1nc(F)nc2n(cnc12)[C@H]1C[C@H](O)[C@@](CO)(O1)C#C
Formula: C12H12FN5O3
Pathway: Microbiology/Virology|||Proteases/Proteasome
Target: HIV Protease|||Reverse Transcriptase
Receptor: N/A
Bioactivity: Islatravir is an effective anti-HIV-1 agent. It acts as a nucleoside reverse transcriptase inhibitor (EC50s: 0.068 nM, 3.1 nM, and 0.15 nM for HIV-1 (WT), HIV-1 (M184V), HIV-1 (MDR), respectively).
Molecular Weight: 293, 258