Product Overview
JKC363 | TP2011 | TargetMol Chemicals
CAS: 436083-30-6
Smiles:
Formula: C69H91N19O16S2
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 0.5 and 44.9 nM at MC4 and MC3 respectively) that antagonizes the effects of α-MSH. Suppresses thyrotropin-releasing hormone (TRH) release, attenuates food intake and reduces formalin-induced pain in vivo.
Molecular Weight: 1506, 72