Product Overview
K-252a | T15636 | TargetMol Chemicals
CAS: 99533-80-9
Smiles: [H][C@]12C[C@](O)(C(=O)OC)[C@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13
Formula: C27H21N3O5
Pathway: Others
Target: Others
Receptor: N/A
Bioactivity: K-252a is a staurosporine analog isolated from Nocardiopsis sp. soil fungi. K-252a inhibits protein kinase (IC50: 470 nM, 140 nM, 270 nM, and 1.7 nM for PKC, PKA, Ca2+/calmodulin-dependent kinase type II, and phosphorylase kinase, respectively).
Molecular Weight: 467, 481
