Product Overview
K 41498 aceate | TP2009L | TargetMol Chemicals
CAS: 0
Smiles:
Formula: N/A
Pathway: GPCR/G Protein
Target: CRFR
Receptor: N/A
Bioactivity: K41498 acetate, an analogues of antisauvagine-30 (aSvg-30), inhibits sauvagine-stimulated cAMP accumulation in hCRF2α- and hCRF2β-expressing cells. K41498 acetate is a potent and highly selective antagonist CRF2 receptor with Ki values of 0.66 nM, 0.62 nM and 425 nM for human CRF2α, CRF2β and CRF1 receptors respectively.
Molecular Weight: N/A