Product Overview
Kuwanon H | TN1849 | TargetMol Chemicals
CAS: 76472-87-2
Smiles: CC(C)=CCc1c(O)ccc(C(=O)[C@H]2[C@@H](CC(C)=C[C@@H]2c2c(O)cc(O)c3c2oc(c(CC=C(C)C)c3=O)-c2ccc(O)cc2O)c2ccc(O)cc2O)c1O
Formula: C45H44O11
Pathway: Endocrinology/Hormones|||GPCR/G Protein
Target: GPR|||Bombesin Receptor
Receptor: N/A
Bioactivity: Kuwanon H is a specific antagonist for the gastrin-releasing peptide (GRP) -preferring receptor with Ki values of 290 nM and can be useful for studying the physiological and pathological role of GRP. Kuwanon H is a potent non-peptide bombesin receptor antagonist.
Molecular Weight: 760, 836
