Product Overview
L-371, 257 | T15682 | TargetMol Chemicals
CAS: 162042-44-6
Smiles: COc1cc(OC2CCN(CC2)C(C)=O)ccc1C(=O)N1CCC(CC1)N1C(=O)OCc2ccccc12
Formula: C28H33N3O6
Pathway: Others
Target: Others
Receptor: N/A
Bioactivity: L-371, 257 is a non-blood-brain barrier penetrant and competitive antagonist of oxytocin receptor (pA2=8.4). It also has high affinity at both the oxytocin receptor (Ki=19 nM) and the vasopressin V1a receptor (Ki=3.7 nM).
Molecular Weight: 507, 587
