Product Overview
Linopirdine | T15758 | TargetMol Chemicals
CAS: 105431-72-9
Smiles: O=C1N(c2ccccc2C1(Cc1ccncc1)Cc1ccncc1)c1ccccc1
Formula: C26H21N3O
Pathway: Membrane transporter/Ion channel
Target: Potassium Channel|||TRP/TRPV Channel
Receptor: N/A
Bioactivity: Linopirdine is a TRPV1 agonist. Linopirdine is an orally active and selective M-type K+ current (IM; Kv7; KCNQ Channels) inhibitor (IC50: 2.4 μM). Linopirdine is a cognitive enhancer. It acts by stimulating release of acetylcholine and other neurotransmitters.Linopirdine is a putative cognition-enhancing drug that increases acetylcholine release in rat brain tissue.
Molecular Weight: 391, 474
