Product Overview
Lintitript | T15759 | TargetMol Chemicals
CAS: 136381-85-6
Smiles: OC(=O)Cn1c(cc2ccccc12)C(=O)Nc1nc(cs1)-c1ccccc1Cl
Formula: C20H14ClN3O3S
Pathway: GPCR/G Protein
Target: cholecystokinin
Receptor: N/A
Bioactivity: Lintitript is an orally active, competitive, and non-peptide cholecystokinin (CCK1) receptor antagonist (EC50: 6 nM; Ki: 0.2 nM). Lintitript shows > 33-fold selectivity more selective for CCK1 than CCK2 receptors (EC50: 200 nM).
Molecular Weight: 411, 86