Product Overview
lumateperone Tosylate | TQ0084 | TargetMol Chemicals
CAS: 1187020-80-9
Smiles: CC1=CC=C(C=C1)S(O)(=O)=O.[H][C@]12CCN(CCCC(=O)C3=CC=C(F)C=C3)C[C@@]1([H])C1=C3N2CCN(C)C3=CC=C1
Formula: C31H36FN3O4S
Pathway: GPCR/G Protein|||Neuroscience
Target: Dopamine Receptor|||5-HT Receptor
Receptor: N/A
Bioactivity: Lumateperone Tosylate is a 5-HT2A receptor antagonist (Ki: 0.54 nM), a SERT blocker (Ki: 61 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki: 32 nM).
Molecular Weight: 565, 7
