Product Overview
LY2922470 | T15810 | TargetMol Chemicals
CAS: 1423018-12-5
Smiles: COc1cccc2CCCN(Cc3ccc(COc4ccc(cc4)[C@H](CC(O)=O)C#CC)s3)c12
Formula: C28H29NO4S
Pathway: Endocrinology/Hormones|||GPCR/G Protein
Target: GPR
Receptor: N/A
Bioactivity: LY2922470 is a potent, selective G protein-coupled receptor 40 (GPR40) agonist, with EC50s of 7 nM for human GPR40, 1 nM for mouse GPR40 and 3 nM for rat GPR40, respectively. LY2922470 reduces glucose levels along and increases insulin and GLP-1 significantly.
Molecular Weight: 475, 6