Lys-[Des-Arg9]Bradykinin acetate | TP1918L1

Lys-[Des-Arg9]Bradykinin acetate | TP1918L1 | TargetMol Chemicals

CAS: TP1918L1

Smiles: [H]N[C@H](C(N[C@H](C(N1CCC[C@H]1C(N2CCC[C@H]2C(NCC(N[C@H](C(N[C@H](C(N3CCC[C@H]3C(N[C@H](C(O)=O)CC4=CC=CC=C4)=O)=O)CO)=O)CC5=CC=CC=C5)=O)=O)=O)=O)CCCNC(N)=N)=O)CCCCN.CC(O)=O

Formula: C52H77N13O13

Pathway: GPCR/G Protein

Target: Bradykinin Receptor

Receptor: N/A

Bioactivity: Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripheral vascular resistance in vivo. 16-fold more potent than [Des-Arg9]-Bradykinin.

Molecular Weight: 1092, 27