[Lys5, MeLeu9, Nle10]-NKA(4-10) | TP1883

[Lys5, MeLeu9, Nle10]-NKA(4-10) | TP1883 | TargetMol Chemicals

CAS: 137565-28-7

Smiles: CCCC[C@H](NC(=O)[C@H](CC(C)C)N(C)C(=O)CNC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](N)CC(O)=O)C(C)C)C(N)=O

Formula: C39H65N9O9

Pathway: GPCR/G Protein|||Neuroscience

Target: Neurokinin receptor

Receptor: N/A

Bioactivity: Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).

Molecular Weight: 804, 003