Product Overview
MK-8617 | T4106 | TargetMol Chemicals
CAS: 1187990-87-9
Smiles: COc1ccc(cc1)C(NC(=O)c1cnc([nH]c1=O)-c1cccnn1)c1ccc(OC)cc1
Formula: C24H21N5O4
Pathway: Chromatin/Epigenetic|||Metabolism
Target: HIF/HIF Prolyl-Hydroxylase
Receptor: N/A
Bioactivity: MK-8617 is an orally available HIF PHD1 3 pan-inhibitor, inhibiting PHD1/2/3 (IC50: 1.0/1.0/14 nM).
Molecular Weight: 443, 463
