Product Overview
MM 54 | TP2001 | TargetMol Chemicals
CAS: 1313027-43-8
Smiles:
Formula: C70H121N29O15S4
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: Potent apelin receptor antagonist (Ki = 82 nM; IC50 = 93 nM). Antagonizes the inhibitory affect of [Pyr1]-Apelin-13 on forskolin-induced cAMP accumulation in CHO-K1-APJ cells. Recuces tumor expansion and lengthens survival time in a mouse xenograft model of glioblastoma.
Molecular Weight: 1737, 15
