Product Overview
MRS 1523 | T16135 | TargetMol Chemicals
CAS: 212329-37-8
Smiles: CCCOC(=O)c1c(CCC)c(C(=O)SCC)c(CC)nc1-c1ccccc1
Formula: C23H29NO3S
Pathway: Others
Target: Others
Receptor: N/A
Bioactivity: MRS 1523 can exert an antihyperalgesic effect through N-type Ca channel block and action potential inhibition in isolated rat dorsal root ganglion (DRG) neurons. MRS 1523 is an effective and selective adenosine A3 receptor antagonist Ki: 18.9 nM and 113 nM for human and rat A3 receptors, respectively). In rat this corresponds to selectivities of 140- and 18-fold vs A1 and A2A receptors, respectively.
Molecular Weight: 399, 55
