Product Overview
MRS2179 | T28099 | TargetMol Chemicals
CAS: 101204-49-3
Smiles: CNc1ncnc2n(cnc12)C1CC(OP(O)([O-])=O)C(COP(O)([O-])=O)O1
Formula: C11H15N5O9P2
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: MRS2179 is a competitive P2Y1 receptor antagonist (Kb = 100 nM) with no appreciable activity at P2Y2, P2Y4, or P2Y6 at concentrations up to 30 µM, or at P2Y12 and P2Y13. It inhibits ADP-induced platelet shape change and aggregation (pA2 = 6.55) in vitro and prolongs bleeding time in rats and mice compared to controls.
Molecular Weight: 423, 216
