Product Overview
MSG606 | TP2002 | TargetMol Chemicals
CAS: 1416983-77-1
Smiles:
Formula: C62H82N20O13S
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: Potent human MC1 receptor antagonist (IC50 = 17 nM). Also partial agonist at human MC3 and MC5 receptors (EC50 values are 59 and 1300 nM, respectively). Exhibits binding affinity for A375 melanoma cells in vitro. Reverses morphine-induced hyperalgesia in female mice, with no effect in male mice. γMSH analog.
Molecular Weight: 1347, 51