Product Overview
N-Desalkylflurazepam | T40366 | TargetMol Chemicals
CAS: 2886-65-9
Smiles: Fc1ccccc1C1=NCC(=O)Nc2ccc(Cl)cc12
Formula: C15H10ClFN2O
Pathway: Membrane transporter/Ion channel|||Metabolism
Target: Calcium Channel
Receptor: N/A
Bioactivity: N-Desalkylflurazepam (Norfludiazepam) is a long-acting metabolite of benzodiazepine compounds, such as Flurazepam. N-Desalkylflurazepam inhibits L-type voltage-gated calcium channels with IC 50 values of 55 μM and 37 μM for Ca v 1.2 and Ca v 1.3, respectively [1] [2] .
Molecular Weight: 288, 71