Product Overview
Napamezole | T28131 | TargetMol Chemicals
CAS: 91524-14-0
Smiles: C(C1=NCCN1)C1=Cc2ccccc2CC1
Formula: C14H16N2
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: Napamezole is an α2 adrenergic receptor antagonist. Napamezole antagonizes methoxamine-induced contractions (alpha-1) of the rat vas deferens with a Kb of 135 nM. Napamezole reverses clonidine-induced decreased in twitch height in the electrically stimulated rat vas deferens.
Molecular Weight: 212, 296