Opiranserin hydrochloride | T9833

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TMC-T9833
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Product Overview

Opiranserin hydrochloride | T9833 | TargetMol Chemicals

CAS: 1440796-75-7

Smiles: O=C(NCC1(N(C)C)CCOCC1)C2=CC(OC)=C(OCCCC)C(OC)=C2.[H]Cl

Formula: C21H35ClN2O5

Pathway: GPCR/G Protein|||Membrane transporter/Ion channel|||Neuroscience

Target: P2X Receptor|||GlyT|||5-HT Receptor

Receptor: N/A

Bioactivity: Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM, respectively. It shows antagonistic activity on rP2X3 (IC50=0.87 μM). It is development as an injectable agent for the treatment of postoperative pain.

Molecular Weight: 430, 97

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