Product Overview
Org 25543 hydrochloride | T22126 | TargetMol Chemicals
CAS: 495076-64-7
Smiles: Cl.COc1cc(cc(OC)c1OCc1ccccc1)C(=O)NCC1(CCCC1)N(C)C
Formula: N/A
Pathway: Neuroscience
Target: GlyT
Receptor: N/A
Bioactivity: Org 25543 hydrochloride is a potent and selective glycine transporter type 2 (GlyT2) inhibitor (IC50 = 16 nM for hGlyT2). Displays no activity at GlyT1 or 56 other common biological targets (≥ 100 μM), in a glycine uptake assay in CHO cells.
Molecular Weight: 448, 983
