Product Overview
OSMI-1 | T16409 | TargetMol Chemicals
CAS: 1681056-61-0
Smiles: COc1ccccc1[C@@H](NS(=O)(=O)c1ccc2[nH]c(=O)ccc2c1)C(=O)N(Cc1ccco1)Cc1cccs1
Formula: C28H25N3O6S2
Pathway: Metabolism|||Others
Target: Others|||Acyltransferase
Receptor: N/A
Bioactivity: OSMI-1 inhibits protein O-linked N-acetylglucosamine (O-GlcNAcylation) in several mammalian cell lines without qualitatively altering cell surface N- or O-linked glycans. OSMI-1 is a cell-permeable O-GlcNAc transferase (OGT) inhibitor (IC50: 2.7 μM).
Molecular Weight: 563, 64
