Product Overview
PD 128042 | T22665 | TargetMol Chemicals
CAS: 114289-47-3
Smiles: CCCCCCCCCCC(C)(C)C(=O)Nc1c(OC)cc(OC)cc1OC
Formula: C23H39NO4
Pathway: Metabolism
Target: Acyltransferase
Receptor: N/A
Bioactivity: CI 976 is a potent orally active and selective ACAT inhibitor(IC50: 73 nM) and a potent lysophospholipid acyltransferase(LPAT) inhibitor. CI 976 inhibits Golgi-associated LPAT activity (IC50: 15 μM) and multiple membrane trafficking steps.
Molecular Weight: 393, 568
