Product Overview
PF-04628935 | T28366 | TargetMol Chemicals
CAS: 1383719-97-8
Smiles: Cc1cn2cc(CC(=O)N3CCC4(CN(Cc5ccc(cc5Cl)-n5nccn5)C4)CC3)nc2s1
Formula: C24H26ClN7OS
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: PF-04628935 is a potent antagonist/inverse agonist of the ghrelin receptor, growth hormone secretagogue receptor 1a (GHS-R1a) with an IC50 of 4.6 nM. PF-04628935 is orally bioavailable and brain penetrant.
Molecular Weight: 496, 03
