PF-05105679 | T16483

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€210.00 - €1,812.00
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TMC-T16483
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Product Overview

PF-05105679 | T16483 | TargetMol Chemicals

CAS: 1398583-31-7

Smiles: C[C@@H](N(Cc1cccc(c1)C(O)=O)C(=O)c1cnc2ccccc2c1)c1ccc(F)cc1

Formula: C26H21FN2O3

Pathway: Membrane transporter/Ion channel

Target: TRP/TRPV Channel

Receptor: N/A

Bioactivity: PF-05105679 is a selective TRPM8 antagonist (IC50 = 103 nM). PF-05105679 can be used in research on cold-related pain.

Molecular Weight: 428, 463

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