Product Overview
Pitstop2 | T9063 | TargetMol Chemicals
CAS: 1332879-52-3
Smiles: O=C1N=C(S/C1=C/C2=CC=C(C=C2)Br)NS(=O)(C3=CC=CC4=C3C=CC=C4)=O
Formula: C20H13BrN2O3S2
Pathway: Microbiology/Virology|||Proteases/Proteasome
Target: HIV Protease
Receptor: N/A
Bioactivity: Pitstop2 is a selective inhibitor of amphiphysin association of clathrin terminal domain with an IC50 value of 12 Ī¼M. Pitstop2 acutely interferes with receptor-mediated endocytosis, entry of HIV, and synaptic vesicle recycling.
Molecular Weight: 473, 36