Product Overview
PRX-08066 Maleic acid | T6959 | TargetMol Chemicals
CAS: 866206-55-5
Smiles: OC(=O)\C=C/C(O)=O.Fc1ccc(CN2CCC(CC2)Nc2ncnc3sc(Cl)cc23)cc1C#N
Formula: C23H21ClFN5O4S
Pathway: GPCR/G Protein|||Neuroscience
Target: 5-HT Receptor
Receptor: N/A
Bioactivity: PRX-08066 Maleic acid is a selective 5-HT2B receptor antagonist with IC50 of 3.4 nM, prevents the severity of pulmonary arterial hypertension in the MCT rat model. Phase 2.
Molecular Weight: 517, 96
