Product Overview
R 892 | TP2126 | TargetMol Chemicals
CAS: 229030-05-1
Smiles:
Formula: C58H83N13O12
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: Potent and selective bradykinin B1 receptor antagonist (ID50 values are 2.8 and > 600 nM at B1 and B2 receptors respectively). Exhibits no intrinsic agonist activity and is resistant to aminopeptidase and kininase II (ACE) cleavage. Displays hypertensive activity in vivo.
Molecular Weight: 1154, 37
