Product Overview
Regadenoson | T2671 | TargetMol Chemicals
CAS: 313348-27-5
Smiles: CNC(=O)c1cnn(c1)-c1nc(N)c2ncn([C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1
Formula: C15H18N8O5
Pathway: GPCR/G Protein|||Neuroscience
Target: Adenosine Receptor
Receptor: N/A
Bioactivity: Regadenoson is an adenosine derivative and selective A2A adenosine receptor agonist with coronary vasodilating activity. Upon administration, regadenoson selectively binds to and activates the A2A adenosine receptor, which induces coronary vasodilation. This leads to an increase in coronary blood flow and enhances myocardial perfusion. Compared to adenosine, regadenoson has a longer half-life and shows higher selectivity towards the A2A adenosine receptor. This agent is a very weak agonist for the A1 adenosine receptor and has negligible affinity for the A2B and A3 adenosine receptors.
Molecular Weight: 390, 36
