Reldesemtiv | T16728

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TMC-T16728
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Product Overview

Reldesemtiv | T16728 | TargetMol Chemicals

CAS: 1345410-31-2

Smiles: NC(=O)c1ccn(c1)-c1cnc(NC[C@@]2(C[C@H](F)C2)c2ncccc2F)nc1

Formula: C19H18F2N6O

Pathway: Others

Target: Others

Receptor: N/A

Bioactivity: Reldesemtiv is a selective and next-generation fast skeletal muscle troponin activator. Reldesemtiv selectively activates fast skeletal myofibrils (EC50: 3.4 μM). Reldesemtiv enhances exercise performance in a heart failure model.

Molecular Weight: 384, 391

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