Product Overview
Siponimod | T6403 | TargetMol Chemicals
CAS: 1230487-00-9
Smiles: CCc1cc(ccc1CN1CC(C1)C(O)=O)C(\C)=N\OCc1ccc(C2CCCCC2)c(c1)C(F)(F)F
Formula: C29H35F3N2O3
Pathway: GPCR/G Protein
Target: S1P Receptor|||LPL Receptor
Receptor: N/A
Bioactivity: BAF312 (Siponimod), a next-generation S1P receptor modulator, is specific for S1P1 and S1P5 receptors with EC50 of 0.39 nM and 0.98 nM, respectively. The specificity of BAF312 for S1P1 and S1P5 receptors exhibits >1000-fold over S1P2, S1P3 and S1P4 receptors.
Molecular Weight: 516, 605
