SR1664 | T23389

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€259.00 - €3,714.00
SKU:
TMC-T23389
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Product Overview

SR1664 | T23389 | TargetMol Chemicals

CAS: 1338259-05-4

Smiles: [H][C@@](C)(\N=C(/O)c1ccc2n(Cc3ccc(cc3)-c3ccccc3C(O)=O)c(C)c(C)c2c1)c1ccc(cc1)N(=O)=O

Formula: C33H29N3O5

Pathway: DNA Damage/DNA Repair|||Metabolism

Target: PPAR

Receptor: N/A

Bioactivity: SR1664 is a potent and selective PPARγ inhibitor with potential antidiabetic activity. SR1664 binds to PPARγ and potently inhibits Cdk5-mediated PPARγ phosphorylation (IC50 = 80 nM; Ki = 28.67 nM) without exhibiting PPARγ agonist activity.

Molecular Weight: 547, 611

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