Product Overview
Talabostat mesylate | T4042 | TargetMol Chemicals
CAS: 150080-09-4
Smiles: CS(O)(=O)=O.CC(C)[C@H](N)C(=O)N1CCC[C@H]1B(O)O
Formula: C10H23BN2O6S
Pathway: Proteases/Proteasome|||Ubiquitination
Target: Proteasome|||DPP-4
Receptor: N/A
Bioactivity: Talabostat mesylate is an orally active, selective inhibitor of dipeptidyl peptidases IV (DPP4, IC50: 0.18 nM), including tumor-associated fibroblast activation protein. This agent may also stimulate the production of colony stimulating factors, such as granulocyte colony-stimulating factor (G-CSF), resulting in the stimulation of hematopoiesis.
Molecular Weight: 310, 17
