Product Overview
Tegoprazan | T17030 | TargetMol Chemicals
CAS: 942195-55-3
Smiles: CN(C)C(=O)c1cc(O[C@H]2CCOc3cc(F)cc(F)c23)c2nc(C)[nH]c2c1
Formula: C20H19F2N3O3
Pathway: Membrane transporter/Ion channel
Target: ATPase|||Proton pump
Receptor: N/A
Bioactivity: Tegoprazan is a potassium-competitive acid blocker and is a potent, oral active, and highly selective inhibitor of gastric H+/K+-ATPase. That could control gastric acid secretion and motility (IC50: ranging from 0.29-0.52 μM for porcine, canine, and human H+/K+-ATPases in vitro).
Molecular Weight: 387, 387