Product Overview
Timapiprant sodium | T17099 | TargetMol Chemicals
CAS: 950688-14-9
Smiles: Cc1c(Cc2ccc3ccccc3n2)c2cc(F)ccc2n1CC(=O)O[Na]
Formula: C21H16FN2NaO2
Pathway: Others
Target: Others
Receptor: N/A
Bioactivity: Timapiprant sodium inhibits mast cell activation of Th2 lymphocytes and eosinophils. Timapiprant sodium is a potent and selective D prostanoid receptor 2 antagonist. Timapiprant sodium potently displaces [3H] PGD2 from human recombinant DP2 (Ki=13 nM), rat recombinant DP2 (Ki=3 nM), human native DP2 (Ki=4 nM).
Molecular Weight: 370, 359
