Product Overview
Tonapofylline | T17117 | TargetMol Chemicals
CAS: 340021-17-2
Smiles: CCCn1c2nc([nH]c2c(=O)n(CCC)c1=O)C12CCC(CCC(O)=O)(CC1)CC2
Formula: C22H32N4O4
Pathway: Others
Target: Others
Receptor: N/A
Bioactivity: Tonapofylline is an orally active and selective adenosine A1 receptor antagonist (Ki: 7.4 nM for human adenosine A1 receptor (hA1)). It shows 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor.
Molecular Weight: 416, 522