Product Overview
Torcetrapib | T2499 | TargetMol Chemicals
CAS: 262352-17-0
Smiles: FC(F)(F)c1cc2c(N([C@@H](C[C@@H]2N(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)OC)CC)C(=O)OCC)cc1
Formula: C26H25F9N2O4
Pathway: Metabolism
Target: CETP
Receptor: N/A
Bioactivity: Torcetrapib is a cholesteryl ester transfer protein (CETP) inhibitor that reduces the heterotypic transfer of cholesteryl ester from HDL to LDL and/or VLDL. Torcetrapib failed in phase III trials due to excess deaths.
Molecular Weight: 600, 47