Product Overview
TPOP146 | T17147 | TargetMol Chemicals
CAS: 2018300-62-2
Smiles: CCC(=O)N1CCOc2c(C1)cc(cc2C(=O)N[C@H]1CCCN(C)C1)-c1cc(OC)cc(OC)c1
Formula: C27H35N3O5
Pathway: Chromatin/Epigenetic
Target: Epigenetic Reader Domain
Receptor: N/A
Bioactivity: TPOP146 is a selective CBP/P300 benzoxazepine bromodomain inhibitor (Kd: 134 nM and 5.02 Ī¼M for CBP and BRD4).
Molecular Weight: 481, 593