Product Overview
UR-3216 | T29074 | TargetMol Chemicals
CAS: 220386-65-2
Smiles: CCOC(=O)Cn1cc2CN(CCc2n1)C(=O)[C@H](Cc1ccc(cc1)[N+]([O-])=O)NC(=O)c1ccc(cc1)C(\N)=N\O
Formula: C27H29N7O7
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: UR-3216, a prodrug, is a selective and orally active platelet surface glycoprotein (GPIIb/IIIa) receptor antagonist. UR-3216 is the very tight binding of its active metabolite to platelets (Ki for resting platelets is < 1 nM). UR-2992, the active form of UR-3216, binds to platelets for a long period of time, while the unbound drug is rapidly cleared.
Molecular Weight: 563, 571
