Product Overview
Urantide | TP2106 | TargetMol Chemicals
CAS: 669089-53-6
Smiles:
Formula: C51H66N10O12S2
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: Selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acetylcholine-induced relaxation. Behaves as a partial agonist in a calcium mobilization assay (in CHO cells expressing hUT receptors).
Molecular Weight: 1075, 26
