Product Overview
VU0529331 | T17246 | TargetMol Chemicals
CAS: 1286725-49-2
Smiles: Cc1ccc(cc1C)-n1nc2CN(Cc2c1-n1cccc1)C(=O)c1cnccn1
Formula: C22H20N6O
Pathway: Others
Target: Others
Receptor: N/A
Bioactivity: VU0529331 is a modestly selective non-GIRK1-containing G protein-gated, inwardly-rectifying, potassium channel activator (EC50s: 5.1 μM and 5.2 μM for GIRK2 and GIRK1/2 in HEK293 cells, respectively). It is also effective on the GIRK4 homomeric channel.
Molecular Weight: 384, 443