WDR5-IN-1 | T13334

WDR5-IN-1 | T13334 | TargetMol Chemicals

CAS: 2408842-51-1

Smiles: COc1cc(CN2CCc3c(cc(Cn4ccn(C)c4=N)cc3-c3ccc(F)cc3C)C2=O)cc(OC)c1

Formula: C30H31FN4O3

Pathway: Others

Target: Others

Receptor: N/A

Bioactivity: WDR5-IN-1 is a potent and selective inhibitor of WD repeat domain 5 (WDR5) (Kd <0.02 nM), and also inhibits MLL1 histone methyltransferase (HMT) activity (IC50: 2.2 nM).

Molecular Weight: 514, 601