Product Overview
Y06137 | T13363 | TargetMol Chemicals
CAS: 2226534-49-0
Smiles: CC1=NOC(C1=C2)=CC=C2C3=NC(C=C4)=C(N3CC5CCCCC5)C=C4N6CCOC[C@@H]6C
Formula: C27H32N4O2
Pathway: Chromatin/Epigenetic|||Cytoskeletal Signaling
Target: Epigenetic Reader Domain|||PKC
Receptor: N/A
Bioactivity: Y06137 is an effective and selective BET inhibitor with a Kd of 81 nM for BRD4(1) bromodomain. Y06137 can be used for research on the treatment of castration-resistant prostate cancer.
Molecular Weight: 444, 57