Product Overview
Zaldaride maleate | T17282 | TargetMol Chemicals
CAS: 109826-27-9
Smiles: OC(=O)\C=C/C(O)=O.CC1(CN2CCC(CC2)n2c3ccccc3[nH]c2=O)OCc2ccccc2-n2cccc12
Formula: C30H32N4O6
Pathway: Others
Target: Others
Receptor: N/A
Bioactivity: Zaldaride maleate inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity (IC50: 3.3 nM). Zaldaride maleate is an effective and selective inhibitor of calmodulin. Zaldaride maleate prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+, and K+ currents in PC12 cells and inhibits nAChR.
Molecular Weight: 544, 608
