Product Overview
Ac-RYYRIK-NH2 acetate | TP1940L1 | TargetMol Chemicals
CAS: TP1940L1
Smiles: NCCCC[C@@H](C(N)=O)NC([C@H]([C@@H](C)CC)NC([C@H](CCCNC(N)=N)NC([C@H](CC1=CC=C(O)C=C1)NC([C@H](CC2=CC=C(O)C=C2)NC([C@H](CCCNC(N)=N)NC(C)=O)=O)=O)=O)=O)=O.CC(O)=O
Formula: C46H74N14O11
Pathway: Endocrinology/Hormones|||GPCR/G Protein|||Neuroscience
Target: Opioid Receptor
Receptor: N/A
Bioactivity: Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity. Ac-RYYRIK-NH2 acetate is a partial agonist on ORL1 transfected in CHO cells, antagonizes the stimulation of [35S]-GTPgammaS binding to G proteins by noc/OFQ in membranes and sections of rat brain.
Molecular Weight: 999, 17
