Product Overview
AdTx1 | TP2086 | TargetMol Chemicals
CAS: TP2086
Smiles:
Formula: C310H481N87O100S8
Pathway: N/A
Target: N/A
Receptor: N/A
Bioactivity: Selective, high affinity, non-competitive α1A adrenoceptor antagonist (Ki = 0.35 nM). Exhibits no significant activity against a range of other GPCRs, including α2A, β1 and β2 adrenoceptors. Antagonizes effects of phenylephrine on isolated rabbit prostate muscle in vitro and on intra-urethral pressure in rats.
Molecular Weight: 7283, 22