Product Overview
AM251 | T1915 | TargetMol Chemicals
CAS: 183232-66-8
Smiles: Cc1c(nn(c1-c1ccc(I)cc1)-c1ccc(Cl)cc1Cl)C(=O)NN1CCCCC1
Formula: C22H21Cl2IN4O
Pathway: Endocrinology/Hormones|||GPCR/G Protein
Target: Cannabinoid Receptor|||GPR
Receptor: N/A
Bioactivity: AM251 is a effective CB1 receptor antagonist (IC50/Ki: 8 /7.49 nM) that displays 306-fold selectivity over CB2 receptors; also effective GPR55 agonist (EC50: 39 nM).
Molecular Weight: 555, 24