CGP 57380 | T6440

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€170.00 - €422.00
SKU:
TMC-T6440
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Product Overview

CGP 57380 | T6440 | TargetMol Chemicals

CAS: 522629-08-9

Smiles: Nc1ncnc2[nH]nc(Nc3ccc(F)cc3)c12

Formula: C11H9FN6

Pathway: Apoptosis|||MAPK

Target: Apoptosis|||MNK

Receptor: N/A

Bioactivity: CGP 57380 is a potent MNK1 inhibitor with IC50 of 2.2 μM, exhibiting no inhibitory activity on p38, JNK1, ERK1 and -2, PKC, or c-Src-like kinases.

Molecular Weight: 244, 233

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