Product Overview
CPI-169 racemate | T6809 | TargetMol Chemicals
CAS: 1450655-76-1
Smiles: CCS(=O)(=O)N1CCC(CC1)C(C)n1c(C)c(C(=O)NCc2c(OC)cc(C)[nH]c2=O)c2ccccc12
Formula: C27H36N4O5S
Pathway: Chromatin/Epigenetic
Target: Epigenetic Reader Domain|||Histone Methyltransferase
Receptor: N/A
Bioactivity: CPI-169 is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively.
Molecular Weight: 528, 67
